产品名称

Squarunkin A

产品货号

Axon 2778 CAS [2101958-02-3] MF C25H32F3N5O4MW 523.55 Purity: 99% Soluble in DMSO Description Squarunkin A selectively inhibits the binding of a myristoylated peptide representing the N-terminus of Src kinase to UNC119A with an IC50 value of 10 nM. It binds to UNC119 proteins in cell lysate and interferes with the activation of Src kinase. KEYWORDS: Squarunkin A | supplier | UNC119–cargo interaction inhibitor | Squarunkin-A | CAS [2101958-02-3] | Non Selective | SRC | Inhibitor | Enzymes | Myristoyl

产品价格

现货询价，电话：010-67529703

产品规格

产品品牌

axonmedchem

产品概述

产品详情

Squarunkin A

Based on 1 reference(s) in Google Scholar 8 10 1

Axon 2778

CAS [2101958-02-3]

MF C25H32F3N5O4
MW 523.55

Purity: 99%
Soluble in DMSO

Squarunkin A

Description

Squarunkin A selectively inhibits the binding of a myristoylated peptide representing the N-terminus of Src kinase to UNC119A with an IC50 value of 10 nM. It binds to UNC119 proteins in cell lysate and interferes with the activation of Src kinase.

T Mejuch et al. Small-Molecule Inhibition of the UNC119-Cargo Interaction. Angew Chem Int Ed Engl. 2017 May 22;56(22):6181-6186.

Selective UNC119–cargo interaction inhibitor

Chemical name

Ethyl 4-(3,4-dioxo-2-(2-(4-(3-(trifluoromethyl)phenyl)piperazin-1-yl)ethylamino)cyclobut-1-enylamino)piperidine-1-carboxylate

Parent CAS No.

[2101958-02-3]

产品资料