产品名称 | BAY-598 |
产品货号 | Axon 2635 CAS [1906919-67-2] MF C22H20Cl2F2N6O3MW 525.34 Purity: 98% Optical purity: 99% e.e. Soluble in DMSO Description BAY-598 is a potent, selective, and cell-active, substrate-competitive inhibitor of SMYD2 (IC50 values of 27 nM and 58 nM for biochemical and cellular activity, respectively). BAY-598 also shows PAR1 antagonism, but there is a greater than 50-fold selectivity for SMYD2 relative to PAR1. KEYWORDS: BAY-598 | supplier | SMYD2 inhibitor | BAY598 | BAY 598 | CAS [1906919-67-2] | Histone | HMTase | Inhibitor | Enzymes | SET | MYND | Protein Methylation | Chemical Probe | Apoptosis | Protein Lysine Methyltransferase | SET and MYND Domain Containing Protein 2 |
产品价格 | 现货询价,电话:010-67529703 |
产品规格 | |
产品品牌 | axonmedchem |
产品概述 | |
产品详情 |
BAY-598Axon 2635 CAS [1906919-67-2] MF C22H20Cl2F2N6O3
DescriptionBAY-598 is a potent, selective, and cell-active, substrate-competitive inhibitor of SMYD2 (IC50 values of 27 nM and 58 nM for biochemical and cellular activity, respectively). BAY-598 also shows PAR1 antagonism, but there is a greater than 50-fold selectivity for SMYD2 relative to PAR1. KEYWORDS: BAY-598 | supplier | SMYD2 inhibitor | BAY598 | BAY 598 | CAS [1906919-67-2] | Histone | HMTase | Inhibitor | Enzymes | SET | MYND | Protein Methylation | Chemical Probe | Apoptosis | Protein Lysine Methyltransferase | SET and MYND Domain Containing Protein 2
Selective inhibitor of SMYD2
Chemical name(S)-N-(1-(N'-Cyano-N-(3-(difluoromethoxy)phenyl)carbamimidoyl)-3-(3,4-dichlorophenyl)-4,5-dihydro-1H-pyrazol-4-yl)-N-ethyl-2-hydroxyacetamide Parent CAS No.[1906919-67-2] |
产品资料 |