| 产品详情 |
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| Product Name | RQ-002303078 |
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| Description | RQ-00203078 is a potent, selective TRPM8 antagonist (IC50 values are 5.3 and 8.3 nM for rat and human channels respectively). Displays >350-fold selectivity for TRPM8 over TRPV4, TRPV1 and TRPA1. RQ-00203078 blocks TRPM8 activity and reduces the invasion potential of oral squamous carcinoma cell lines. RQ-00203078 (RQ) profoundly reduced such agonist-induced cation currents. MW: 554.85. Purity ≥98% by HPLC |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 4-[[[3-Chloro-5-(trifluoromethyl)-2-pyridinyl][[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]benzoic ac |
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| Gene, Accession, CAS # | CAS: 1254205-52-1 |
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| Catalog # | 9636-10 |
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| Order / More Info | RQ-002303078 from BIOVISION, INC. |
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| Product Specific References | n/a |
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