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| Product Name | BRL 54443 |
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| Description | A potent 5-ht1E/1F receptor agonist (pEC50 values are 8.5 and 8.6 respectively). Displays > 30-fold selectivity over other 5-HT and dopamine receptors (pKi values are 8.7. 8.9, 7.2, 6.9, 7.2, 5.9, 7.0, 6.5, < 6, < 6, 6.3 and 6.2 for human 5-HT1E, 1F, 1A, 1B, 1D, 2A, 2B, 2C, 4, 7, D2 and D3 receptors respectively). Induces 5-HT2A receptor-mediated mouse aortic contraction in vitro (pEC50 = 6.52). Active in vivo. MW (observed): 230.31. |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 5-Hydroxy-3-(1-methylpiperidin-4-yl)-1H-indole |
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| Gene, Accession, CAS # | CAS: 57477-39-1 |
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| Catalog # | 1129/10 |
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| Price | |
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| Order / More Info | BRL 54443 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 19649285, 21422162 |
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| 产品资料 |
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