产品详情 |
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Product Name | CI 988 |
Description | Potent and selective CCK2 (CCK-B) receptor antagonist that displays ~ 1600-fold selectivity over CCK1 receptors (IC50 values are 1.7 and 2717 nM for CCK2 and CCK1 respectively). Has negligible affinity at a range of other binding sites (IC50 > 10 μM). Exhibits anxiolytic activity following oral administration. Purity 99%. MW (observed): 614.73 |
Size | 50 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-1-oxo-2-[[(tricyclo[3.3.1.13,7]dec-2-yloxy)carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid. PD 134308 |
Gene, Accession, CAS # | CAS: 130332-27-3 |
Catalog # | 2607/50 |
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Order / More Info | CI 988 from TOCRIS BIOSCIENCE
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Product Specific References | n/a |
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