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| Product Name | INCB 3284 dimesylate |
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| Description | Potent, selective hCCR2 antagonist. Exhibits potent antagonism against monocyte chemoattractant molecule binding to hCCR2 and chemotaxis activity (IC50 values are 3.7 and 4.7 nM respectively). Also displays weak hERG activity; inhibits the hERG potassium current (IC50 = 84μM). Orally bioavailable. Purity 98%. MW (observed): 712.76 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | N-[2-[[(3R)-1-[trans-4-Hydroxy-4-(6-methoxy-3-pyridinyl)cyclohexyl]-3-pyrrolidinyl]amino]-2-oxoethyl]-3-(trifluoromethyl)-benzamide dimethanesulfonate |
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| Gene, Accession, CAS # | CAS: 887401-93-6 |
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| Catalog # | 4306/10 |
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| Price | |
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| Order / More Info | INCB 3284 dimesylate from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 24904083, 25012628, 27216982 |
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