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Product Name | AM 251 |
Description | Potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors. Also potent GPR55 agonist (EC50 = 39 nM) and μ-opioid receptor antagonist (Ki = 251 nM). Fluorescent Form also available.. Purity 99%. MW (observed): 555.24 |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide |
Gene, Accession, CAS # | CAS: 183232-66-8 |
Catalog # | 1117/10 |
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Order / More Info | AM 251 from TOCRIS BIOSCIENCE
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Product Specific References | PubMed: 11454655, 11588122, 11877326, 12578907, 14623770, 15140923, 15155534, 15163690, 15187170, 15249429, 15266010, 15277315, 15277316, 15280536, 15363397, 15451779, 15525762, 15629705, 15673670, 15721795, 15821037, 16025138, 16262678, 16301180, 16331291, 16357196, 16467564, 16513651, 16624937, 16675398, 16705137, 16715117, 16775133, 16988037, 17004927, 17043671, 17045264, 17202425, 17227847, 17289026, 17301239, 17475795, 17486141, 17557913, 17586490, 17652447, 17652632, 17653268, 17684555, 17881527, 18093525, 18156315, 18162180, 18266975, 18335063, 18341994, 18355636, 18469844, 18486111, 18493584, 18552868, 18614676, 18687967, 18695638, 18723035, 18794527, 18846037, 18930826, 18955347, 19091987, 19133994, 19158669, 19284549, 19325030, 19594755, 19666749, 19681872, 19845674, 19906779, 19907129, 20071517, 20074214, 20136841, 20144892, 20174577, 20196921, 20233215, 20305287, 20435001, 20534730, 20590576, 20639875, 20668190, 20718749, 20720126, 20729846, 20884761, 20926585, 20927050, 20955176, 21095576, 21148002, 21177997, 21182571, 21241462, 21439272, 21447623, 21470203, 21755008, 21844187, 21918506, 21937980, 21940435, 21951063, 22031841, 22046372, 22073164, 22139792, 22266354, 22285397, 22291615, 22368777, 22413007, 22428664, 22429826, 22549120, 22553354, 22715379, 22848724, 22913292, 22940464, 22959963, 22989885, 23015449, 23055515, 23139770, 23285225, 23347118, 23394117, 23426383, 23493814, 23675095, 23712280, 23739343, 23806960, 23894352, 23939223, 24030632, 24089517, 24312195, 24324206, 24349109, 24469251, 24589887, 24758718, 24847420, 24899717, 25030704, 25481343, 25505329, 25535367, 25575795, 25653478, 25684407, 25731744, 25830356, 25891347, 25915740, 25943894, 26085115, 26090232, 26092099, 26215450, 26414859, 26482099, 26558388, 26648844, 26671069, 26920222, 27285468, 27418880, 27641813, 28322749, 28479394, 28750085, 28987618, 29237478 |
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