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| Product Name | LY 393558 |
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| Description | Dual 5-HT1B/1D receptor antagonist (pKB values are 9.05 and 8.98 respectively) and 5-HT re-uptake inhibitor (pIC50 = 8.48). Potently antagonizes terminal autoreceptor activity in vitro and increases extracellular 5-HT levels above those evoked by fluoxetine (Cat. No. 0927) in vivo. Also acts as an antagonist at 5-HT2A and 5-HT2B receptors (pKi values are 7.29 and 7.35 respectively). Purity 97%. MW (observed): 546.68 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | 1-[2-[4-(6-Fluoro-1H-indol-3-yl)-3,6-dihydro-1(2H)-pyridinyl]ethyl]-3,4-dihydro-3-(1-methylethyl)-6-(methylsulfonyl)-1H-2,1,3-benzothiadiazine-2,2-dioxide |
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| Gene, Accession, CAS # | CAS: 271780-64-4 |
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| Catalog # | 3350/10 |
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| Price | |
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| Order / More Info | LY 393558 from TOCRIS BIOSCIENCE
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| Product Specific References | n/a |
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| 产品资料 |
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