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| Product Name | Eliprodil |
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| Description | Non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site. Selective for GluN2B (formally NR2B)- over GluN2A (NR2A)- and GluN2C (NR2C)-containing receptors (IC50 values are 1, > 100 and > 100 μM respectively). Also σ1 ligand (Ki = 0.013 μM). Antagonizes neuronal voltage-gated Ca2+ channels and selectively inhibits the rapid component of the delayed rectifier K+ current (IKr). Neuroprotective. Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions. Purity 98%. MW (observed): 347.86 |
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| Size | 10 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | α-(4-Chlorophenyl)-4-[(4-fluorophenyl)methyl]-1-piperidineethanol |
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| Gene, Accession, CAS # | CAS: 119431-25-3 |
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| Catalog # | 2195/10 |
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| Price | |
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| Order / More Info | Eliprodil from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 22197913, 27239788 |
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